Structure and mechanism of mammalian ferroportin

NIH RePORTER · NIH · R01 · $400,000 · view on reporter.nih.gov ↗

Abstract

Project Summary: Ferroportin is the only iron exporter in humans. Mutations in ferroportin cause hemochromatosis. Ferrorpotin is regulated by a peptide hormone hepcidin, which is produced in the liver and inhibits the activity of ferrorportin by inducing endocytosis and by direct inhibition of ferroportin activity. The FPN-hepcidin axis is a potential therapeutic target for normalizing iron homeostasis in hemochromatosis. However, very little is known about how ferroportin recognizes and transport iron and how it interacts with hepcidin. In this study, I will combine structural and functional analyses to understand the mechanism of iron transport and inhibition in ferroportin at the atomic resolution.

Key facts

NIH application ID
10397598
Project number
5R01HL157473-02
Recipient
BAYLOR COLLEGE OF MEDICINE
Principal Investigator
Yaping Pan
Activity code
R01
Funding institute
NIH
Fiscal year
2022
Award amount
$400,000
Award type
5
Project period
2021-05-01 → 2025-04-30