Sex specific epigenetic regulation of colon cancer metastasis

NIH RePORTER · NIH · R01 · $403,649 · view on reporter.nih.gov ↗

Abstract

Colorectal cancer (CRC) is the third leading cause of cancer death in US and is characterized by signature mutations of APC, p53, KRAS, SMAD4, among other genetic alterations. It is well established that male CRC patients have worse prognosis than that of female patients, but the underlying mechanism is largely undefined. Recent efforts in large scale whole genome and whole exome sequencing of metastatic CRC samples have not identified novel metastatic promoting genes suggesting metastatic progression may be largely regulated by epigenetic mechanisms. We have recently established an inducible oncogenic KRas metastatic CRC animal model and employing this model we have identified a male specific Y-chromosome residing gene- KDM5D, as a key regulator of CRC metastatic progression. This discovery is exciting as it connects sex biased CRC progression with an epigenetic regulator that is druggble. In this proposal, we will employ both in vitro and animal models to elucidate the function of KDM5D in CRC progression and define novel therapeutic approach targeting CRC metastasis. To achieve this goal, we propose the following specific aims. 1. Elucidate the role of KDM5D in CRC progression; 2. Define Kras mediated KDM5D upregulation in CRC and KDM5D downstream targets in promoting metastasis; 3. Mechanistic understanding of KDM5D promotion of metastasis in vivo.

Key facts

NIH application ID
10443932
Project number
1R01CA262798-01A1
Recipient
INDIANA UNIVERSITY INDIANAPOLIS
Principal Investigator
Y. Alan Wang
Activity code
R01
Funding institute
NIH
Fiscal year
2022
Award amount
$403,649
Award type
1
Project period
2022-09-06 → 2027-08-31