Optimization of microtubule-stabilizing triazolopyrimidines as therapeutics for Alzheimer's disease and related tauopathies

NIH RePORTER · NIH · U01 · $311,482 · view on reporter.nih.gov ↗

Abstract

Statement of Work Specific activities overseen by the Brunden laboratory include: 1) testing of prodrugs in established HEK293 and neuron microtubule stabilization assays; 2) intravenous and oral pharmacokinetic testing of prodrugs to determine the rate of conversion of prodrugs to the desired active compound; 3) assessment of preferred prodrugs for pharmacodynamic effect in wild-type mice to establish the minimum effective dose and duration of compound effect; and 4) determination of preferred prodrug acute maximum tolerated dose and the no adverse effect dose after 3 weeks of dosing.

Key facts

NIH application ID
10553899
Project number
3U01AG061173-04S1
Recipient
UNIVERSITY OF PENNSYLVANIA
Principal Investigator
KURT R. BRUNDEN
Activity code
U01
Funding institute
NIH
Fiscal year
2022
Award amount
$311,482
Award type
3
Project period
2019-03-01 → 2024-02-29