Developing Selective P-catalysts for Dehydrative Transformations

NIH RePORTER · NIH · F32 · $74,284 · view on reporter.nih.gov ↗

Abstract

PROJECT SUMMARY/ABSTRACT This proposal will elucidate the various steric and electronic parameters of a P-catalyst necessary for enantioinduction in tandem amidation/amide functionalizations through deoxygenative P(III)/P(V) catalysis; an important transformation for the synthesis of biologically active compounds. This proposal will first examine P- catalyzed enantioselective amidations, followed by P-catalyzed enantioretentive amide functionalizations. Finally, these catalysts will be combined for a one-pot synthesis of enantioenriched secondary nitriles from racemic carboxylic acids, a moiety important to the pharmaceutical community. Overall, during this fellowship period I seek to gain expertise in inorganic main-group chemistry, including computational analyses and modern inorganic synthetic techniques. Such skills will complement my existing skillset, creating a strong foundation in catalyst design for my future career goals.

Key facts

NIH application ID
10827018
Project number
1F32GM153091-01
Recipient
MASSACHUSETTS INSTITUTE OF TECHNOLOGY
Principal Investigator
Siraj Zaki Ali
Activity code
F32
Funding institute
NIH
Fiscal year
2024
Award amount
$74,284
Award type
1
Project period
2024-02-01 → 2026-01-31