Total Synthesis of Dodecahedrane via Carbon–Carbon Bond Forming Cascades

NIH RePORTER · NIH · F31 · $43,860 · view on reporter.nih.gov ↗

Abstract

Project Summary/Abstract The chemical synthesis of small molecules continues to be a vital area of research. Such efforts can lead to the development of new and improved methods, provide access to interesting or important scaffolds, and provide fundamental insight into reactivity and synthetic design that, in turn, can enable future research endeavors. This proposal is focused on achieving the total synthesis of the complex molecule dodecahedrane via the development of carbon–carbon bond forming reaction cascades. In Aim 1, a dimeric norbornyl scaffold will be prepared and utilized in an olefin metathesis isomerization reaction. This endeavor will provide access to a late-stage intermediate, while enabling the investigation and development of a unique variant of olefin methathesis for the assembly of molecular complexity. In Aim 2, a symmetrical penta-ene substrate will be synthesized and used in a unique and ambitious poly-ene cyclization, involving all five alkenes, to access dodecahedrane in the final synthetic step.

Key facts

NIH application ID
10848238
Project number
5F31GM148017-02
Recipient
UNIVERSITY OF CALIFORNIA LOS ANGELES
Principal Investigator
Luca McDermott Catena
Activity code
F31
Funding institute
NIH
Fiscal year
2024
Award amount
$43,860
Award type
5
Project period
2023-07-01 → 2025-06-30