Neural Ice Technology for Treatment of Pain

NIH RePORTER · NIH · R44 · $998,787 · view on reporter.nih.gov ↗

Abstract

Total knee arthroplasty (TKA) is one of the most performed orthopedic surgeries to relieve joint pain in patients with end-stage osteoarthritis (OA) or rheumatic arthritis (RA). In the US, over 700,000 TKA procedures are performed annually. To manage TKA pain patients are commonly prescribed opioids, contributing to a spiraling opioid epidemic. The misuse and addiction to opioids is a national public health crisis with an estimated economic burden of $78.5 billion per year. As opioid addiction is now a national health focus, novel non-opioid and non-pharmacological treatments for postoperative pain are a top scientific priority. There is an urgent need for a long-lasting, drug-free means of relieving post-TKA pain–which is the overall goal of this project. Cryoneurolysis is an opioid-sparing, perioperative intervention used to reduce postoperative pain. Current cryoneurolysis methods apply very low-temperature cryoprobes to freeze peripheral nerves, resulting in reversible and long-lasting pain relief. However, due to extremely cold temperatures (–88oC and below) in direct contact with a nerve and surrounding tissues, these methods are not nerve-selective nor easy to administer. They also are not injectable, making the treatments time-consuming and challenging to adopt in clinic. Our initial goal – an easier to use, injectable method of cryoneurolysis to reduce postoperative pain from TKA, significantly reducing or eliminating the use of opioids. We invented a novel injectable and nerve-selective cryoneurolysis method that overcomes the limitations of current options. Neural Ice™ can be injected around sensory peripheral nerves that transmit pain. We have shown in a rat model that injection of our ice-slurry, formulated to bring peri-nerve temperatures to around -5oC, extracts enough thermal energy to reversibly disrupt nerve structure and reduce pain sensation for up to 8 weeks without damage to surrounding tissue. At the end of 2023, we also completed an initial 16-patient feasibility study showing significant pain reduction response with no serious adverse events (See Significance). In response to these findings (pre-clinical and clinical) in October 2023 the FDA granted Brixton Breakthrough Designation. In Phase II, we seek to optimize a clinical use device that produces an injectable, biocompatible, and sterile ice slurry which meets the FDA requirements for an Investigative Device Exemption (IDE) for a pivotal efficacy trial. With our HEAL Phase I grant we generated single-use, terminally sterilized pre-filled syringes that contain on-demand injectable slurry for use at point-of-care facilities. In Phase II we seek to optimize our design for human use (ease, effectiveness, cost, etc.) and test for in-vivo biologic response in rat model. We will also establish manufacturing of human use system & prepare to submit pivotal trial IDE application to the FDA at the end of the funding period. If successful, our study will lead to the development...

Key facts

NIH application ID
11006862
Project number
1R44AR084998-01
Recipient
BRIXTON BIOSCIENCES, INC.
Principal Investigator
Charles Sidoti
Activity code
R44
Funding institute
NIH
Fiscal year
2024
Award amount
$998,787
Award type
1
Project period
2024-08-21 → 2026-07-31