SynerGel: A Novel Tumor Microenvironment-Modulating Hydrogel for Local Immunotherapy

NIH RePORTER · NIH · R01 · $77,282 · view on reporter.nih.gov ↗

Abstract

PROJECT SUMMARY. Conventional multi-modality therapy for Head and Neck Squamous Cell Carcinoma (HNSCC), such as surgery and chemoradiotherapy, can result in off-target effects and often fails to eradicate cancer, resulting in high locoregional and distant recurrence rates. The adverse tumor immune microenvironment (TIME) in HNSCC has been shown to: 1) impair tumor-infiltrating lymphocyte function, 2) decrease the production of effector cytokines, and 3) contain suppressive immunocytes. Thus, there is strong interest in developing strategies to mitigate the suppressive TIME and elicit a strong anti-tumor immune response. A successful immunotherapy approach should also boost immunological memory and thus reduce cancer recurrence. Most HNSCC patients treated with single-agent FDA-approved immunotherapies do not respond, in large part due to the immunosuppressive TIME. A drug delivery innovation that addresses immunotherapy's shortcomings while reducing side effects could significantly impact HNSCC treatment. To overcome these limitations, we propose a novel hydrogel-based platform for spatiotemporal control over the delivery of cytokines, specifically, lnterleukin-2 (IL-2), lnterleukin-12 (IL-12), and lnterleukin-15 (IL-15) to stimulate antitumor effector cells and suppress myeloid-derived suppressive cells (MDSCs). Our L-NIL functionalized multi-domain peptide hydrogel platform (SynerGel) can be injected intratumorally to deliver and release immunomodulators into the TIME locally. We hypothesize the combination of cytokines in our SynerGe/ platform will localize and extend the release of these immunomodulators intratumorally, stimulating anti-tumor effector immunocytes in synergy with the suppression of MDSCs. To investigate this hypothesis, we will evaluate SynerGe/ as an injectable, highly customizable cancer immunotherapy platform able to perform sustained delivery of multiple cytokines to the TIME (Aim 1) and identify specific immune mechanisms contributing to the efficacy of cytokine-releasing SynerGels in the HNSCC tumor microenvironment (Aim 2). We anticipate the combination of cytokines in SynerGel will have controlled release, suppress MDSCs, and stimulate anti-tumor effector immune cells for durable responses. This project offers a biomaterial-based approach to deliver immunotherapeutics to the suppressive TIME in HNSCC. Dr. Simon Young will serve as the primary mentor of the trainee with the co-mentorship of Dr. Mary Cindy Farach-Carson. During graduate degree training, the candidate will meet with mentors regularly, write first-author publications, and present research findings at conferences. This supplement will help the trainee develop scientific and communication skills, leadership qualities, and a deeper understanding of the tumor immune microenvironment in head and neck cancers, aligning with the candidate's goal of becoming an independent translational researcher.

Key facts

NIH application ID
11064107
Project number
3R01DE030140-04S1
Recipient
UNIVERSITY OF TEXAS HLTH SCI CTR HOUSTON
Principal Investigator
Simon Young
Activity code
R01
Funding institute
NIH
Fiscal year
2024
Award amount
$77,282
Award type
3
Project period
2021-07-01 → 2025-04-30