Exploring Peptide Conjugates as Trojan Horse Systems for Drug Design and Discovery

NIH RePORTER · NIH · R01 · $413,897 · view on reporter.nih.gov ↗

Abstract

 DESCRIPTION (provided by applicant): Microcin C7 (McC) is a potent natural product antimicrobial produced by enterobacteria. McC enters the target cell using a "Trojan horse" strategy, in which the active portion of the antibiotic is coupled to a peptide carrier that faciliates import into target cell through active transporters. We have characterized several biosynthetic clusters for that produce the same antibiotic component but with different peptide attachments. Presumably, changes in the peptide allow for import through different transport systems that are specific to different bacterial species. Here we seek to: i. install variations in the peptide carrer allowing the molecule to be taken up by diverse bacteria. ii. re-design the peptide carrier so that it can be more effectively imported into susceptible organisms.

Key facts

NIH application ID
9823840
Project number
5R01AI117210-05
Recipient
UNIVERSITY OF ILLINOIS AT URBANA-CHAMPAIGN
Principal Investigator
Satish K Nair
Activity code
R01
Funding institute
NIH
Fiscal year
2020
Award amount
$413,897
Award type
5
Project period
2015-12-01 → 2020-11-30