Mechanisms of Resistance to mTOR Targeted Therapies

NIH RePORTER · VA · I01 · · view on reporter.nih.gov ↗

Abstract

The broad objective of this proposal is to investigate the intrinsic mechanisms of tumor cell resistance to newly developed mTOR inhibitors such that their future use may be optimized in the clinic. We have identified an alternate mechanism of mRNA translation initiation that is activated upon mTOR inhibitor exposure allowing tumor cell survival in the face of global inhibition of protein synthesis. These experiments will delineate the molecular mechanisms promoting activation of this salvage pathway and will pre-clinically evaluate the repurposing of an FDA-approved drug as a small molecule inhibitor targeting this pathway for synergistic antitumor effects in combination with mTOR inhibitors. We will utilize a combination of genetic and biochemical approaches to address the molecular mechanisms by which the salvage protein synthesis pathway is activated in TOR inhibitor resistant brain cancers. We will utilize mouse models of these diseases to evaluate the efficacy of these inhibitors.

Key facts

NIH application ID
9932900
Project number
5I01BX002665-07
Recipient
VA GREATER LOS ANGELES HEALTHCARE SYSTEM
Principal Investigator
JOSEPH F GERA
Activity code
I01
Funding institute
VA
Fiscal year
2020
Award amount
Award type
5
Project period
2014-07-01 → 2022-06-30