Development of Sulfur-Based Reactions with Translational Applications

NIH RePORTER · NIH · R01 · $113,257 · view on reporter.nih.gov ↗

Abstract

Abstract Synthesis and coupling of hindered and strained functional molecules and bioisosteres represent underdeveloped yet synthetically powerful transformations. This research project is focused on the discovery of both stoichiometric and catalytic sulfur mediated couplings, which might that potentially overcome several limitations often encountered in traditional transition-metal couplings. Our research heavily relies on UPLC analysis and purification because of the reaction development, molecular complexity and unique physical properties of sulfurane, boronates, bicyclo[1.1.1]pentanes, sp3-rich amines and other polar bioactive molecules. The goal of this administrative supplement application is to strengthen the analytical capability of this research program.

Key facts

NIH application ID
11098352
Project number
3R01GM141088-04S1
Recipient
UT SOUTHWESTERN MEDICAL CENTER
Principal Investigator
Tian Qin
Activity code
R01
Funding institute
NIH
Fiscal year
2024
Award amount
$113,257
Award type
3
Project period
2021-04-01 → 2026-03-31