Multimodal Gating Mechanisms of TRPV1 Ion Channels

NIH RePORTER · NIH · R01 · $419,850 · view on reporter.nih.gov ↗

Abstract

Project summary The goal of this proposal is to determine the molecular mechanisms underlying multi-modal gating of the pain-receptor ion channel TRPV1 by interrogating the structural mechanisms for activation by capsaicin, heat, protons, savory compounds, and signaling lipids. We will use tmFRET and computational methods to determine the conformational change induced by each modality and the coupling between modalities.

Key facts

NIH application ID
9843458
Project number
5R01GM125351-03
Recipient
UNIVERSITY OF WASHINGTON
Principal Investigator
Sharona E Gordon
Activity code
R01
Funding institute
NIH
Fiscal year
2020
Award amount
$419,850
Award type
5
Project period
2018-01-01 → 2021-12-31